Aspirina e outros anti-inflamatórios não esteroidais (AINEs) devem ser usados com cuidado, especialmente em pessoas com mais de 60 anos de idade ou aquelas também medicadas com corticosteroides, bifosfonatos ou outros medicamentos antitrombóticos.[24]García Rodríguez LA, Lin KJ, Hernández-Díaz S, et al. Risk of upper gastrointestinal bleeding with low-dose acetylsalicylic acid alone and in combination with clopidogrel and other medications. Circulation. 2011 Mar 15;123(10):1108-15.
https://www.ahajournals.org/doi/10.1161/CIRCULATIONAHA.110.973008?url_ver=Z39.88-2003&rfr_id=ori:rid:crossref.org&rfr_dat=cr_pub%20%200pubmed
http://www.ncbi.nlm.nih.gov/pubmed/21357821?tool=bestpractice.com
[25]Knopp-Sihota JA, Cummings GG, Homik J, et al. The association between serious upper gastrointestinal bleeding and incident bisphosphonate use: a population-based nested cohort study. BMC Geriatr. 2013 Apr 20;13:36.
https://bmcgeriatr.biomedcentral.com/articles/10.1186/1471-2318-13-36
http://www.ncbi.nlm.nih.gov/pubmed/23602075?tool=bestpractice.com
O uso concomitante de um inibidor da bomba de prótons (IBP) demonstrou reduzir o risco de complicações gastrointestinais em pacientes submetidos a uma terapia com aspirina e/ou anticoagulantes orais em longo prazo.[35]Scheiman JM, Devereaux PJ, Herlitz J, et al. Prevention of peptic ulcers with esomeprazole in patients at risk of ulcer development treated with low-dose acetylsalicylic acid: a randomised, controlled trial (OBERON). Heart. 2011 May;97(10):797-802.
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3088470/?tool=pubmed
http://www.ncbi.nlm.nih.gov/pubmed/21415072?tool=bestpractice.com
[36]Kurlander JE, Barnes GD, Fisher A, et al. Association of antisecretory drugs with upper gastrointestinal bleeding in patients using oral anticoagulants: a systematic review and meta-analysis. Am J Med. 2022 Oct;135(10):1231-43.e8.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10031639
http://www.ncbi.nlm.nih.gov/pubmed/35679879?tool=bestpractice.com
[37]Ahn HJ, Lee SR, Choi EK, et al. Protective effect of proton-pump inhibitor against gastrointestinal bleeding in patients receiving oral anticoagulants: a systematic review and meta-analysis. Br J Clin Pharmacol. 2022 Nov;88(11):4676-87.
http://www.ncbi.nlm.nih.gov/pubmed/35921204?tool=bestpractice.com
Os IBPs previnem as úlceras pépticas e as complicações em pessoas que necessitam de terapia com AINE.[38]Yang M, He M, Zhao M, et al. Proton pump inhibitors for preventing non-steroidal anti-inflammatory drug induced gastrointestinal toxicity: a systematic review. Curr Med Res Opin. 2017 Jan 25;33(6):973-80.
http://www.ncbi.nlm.nih.gov/pubmed/28076696?tool=bestpractice.com
No entanto, as diretrizes sugerem considerar uma estratégia de teste e tratamento para o Helicobacter pylori antes de iniciar a terapia em longo prazo com AINEs, uma vez que a erradicação do H pylori demonstrou proteger contra o sangramento da úlcera péptica associada à aspirina.[33]Lanza FL, Chan FK, Quigley EM; Practice Parameters Committee of the American College of Gastroenterology. Guidelines for prevention of NSAID-related ulcer complications. Am J Gastroenterol. 2009 Mar;104(3):728-38.
http://www.ncbi.nlm.nih.gov/pubmed/19240698?tool=bestpractice.com
[39]Hawkey C, Avery A, Coupland CAC, et al. Helicobacter pylori eradication for primary prevention of peptic ulcer bleeding in older patients prescribed aspirin in primary care (HEAT): a randomised, double-blind, placebo-controlled trial. Lancet. 2022 Nov 5;400(10363):1597-606.
https://www.thelancet.com/journals/lancet/article/PIIS0140-6736(22)01843-8/fulltext
http://www.ncbi.nlm.nih.gov/pubmed/36335970?tool=bestpractice.com
A terapia com IBPs pode ser mais efetiva que o misoprostol (um análogo da prostaglandina E1) para a prevenção de úlceras gastrointestinais nas pessoas com prescrição de terapia com AINEs de longa duração.
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Do misoprostol, H2-receptor antagonists, or proton pump inhibitors used for at least 12 weeks prevent upper gastrointestinal ulcers in patients requiring chronic NSAID use?/cca.html?targetUrl=https://cochranelibrary.com/cca/doi/10.1002/cca.430/fullMostre-me a resposta A adesão terapêutica ao misoprostol (particularmente em altas doses) pode ser comprometida por efeitos adversos gastrointestinais, incluindo cólicas abdominais e diarreia.
O uso profilático de um IBP é apropriado para os pacientes em terapia intensiva, que são considerados de alto risco para hemorragia digestiva devido a comorbidades, como doença hepática crônica, ou que tiverem condições como coagulopatia, choque ou doença hepática coexistentes.[34]MacLaren R, Dionne JC, Granholm A, et al. Society of Critical Care Medicine and American Society of Health-System Pharmacists Guideline for the prevention of stress-related gastrointestinal bleeding in critically ill adults. Crit Care Med. 2024 Aug 1;52(8):e421-30.
https://journals.lww.com/ccmjournal/fulltext/2024/08000/society_of_critical_care_medicine_and_american.22.aspx
http://www.ncbi.nlm.nih.gov/pubmed/39007578?tool=bestpractice.com
[40]Cash BD. Evidence-based medicine as it applies to acid suppression in the hospitalized patient. Crit Care Med. 2002 Jun;30(suppl 6):S373-8.
http://www.ncbi.nlm.nih.gov/pubmed/12072665?tool=bestpractice.com
A ventilação mecânica, por si só, não é mais considerada um fator de risco.[34]MacLaren R, Dionne JC, Granholm A, et al. Society of Critical Care Medicine and American Society of Health-System Pharmacists Guideline for the prevention of stress-related gastrointestinal bleeding in critically ill adults. Crit Care Med. 2024 Aug 1;52(8):e421-30.
https://journals.lww.com/ccmjournal/fulltext/2024/08000/society_of_critical_care_medicine_and_american.22.aspx
http://www.ncbi.nlm.nih.gov/pubmed/39007578?tool=bestpractice.com
[41]Mutlu GM, Mutlu EA, Factor P. Prevention and treatment of gastrointestinal complications in patients on mechanical ventilation. Am J Respir Med. 2003;2(5):395-411.
http://www.ncbi.nlm.nih.gov/pubmed/14719992?tool=bestpractice.com
Todos os adultos gravemente enfermos com fatores que provavelmente aumentam o risco de hemorragia digestiva alta relacionada a estresse devem receber um IBP ou um antagonista H2 para prevenir sangramentos.[42]Reynolds PM, MacLaren R. Re-evaluating the utility of stress ulcer prophylaxis in the critically ill patient: a clinical scenario-based meta-analysis. Pharmacotherapy. 2019 Mar;39(3):408-20.
http://www.ncbi.nlm.nih.gov/pubmed/30101529?tool=bestpractice.com
[34]MacLaren R, Dionne JC, Granholm A, et al. Society of Critical Care Medicine and American Society of Health-System Pharmacists Guideline for the prevention of stress-related gastrointestinal bleeding in critically ill adults. Crit Care Med. 2024 Aug 1;52(8):e421-30.
https://journals.lww.com/ccmjournal/fulltext/2024/08000/society_of_critical_care_medicine_and_american.22.aspx
http://www.ncbi.nlm.nih.gov/pubmed/39007578?tool=bestpractice.com
A profilaxia deve ser descontinuada quando a doença crítica não for mais evidente ou o(s) fator(es) de risco não estiverem mais presentes apesar de uma doença crítica em curso.[34]MacLaren R, Dionne JC, Granholm A, et al. Society of Critical Care Medicine and American Society of Health-System Pharmacists Guideline for the prevention of stress-related gastrointestinal bleeding in critically ill adults. Crit Care Med. 2024 Aug 1;52(8):e421-30.
https://journals.lww.com/ccmjournal/fulltext/2024/08000/society_of_critical_care_medicine_and_american.22.aspx
http://www.ncbi.nlm.nih.gov/pubmed/39007578?tool=bestpractice.com
A descontinuação da profilaxia para úlcera por estresse fisiológico antes da transferência para fora da unidade de terapia intensiva é necessária para evitar prescrições inadequadas.[43]Jones CA, Betthauser KD, Lizza BD, et al. Impact of stress ulcer prophylaxis discontinuation guidance in mechanically ventilated, critically ill patients: a pre-post cohort study. Hosp Pharm. 2022 Aug;57(4):510-7.
https://pmc.ncbi.nlm.nih.gov/articles/PMC9310319
http://www.ncbi.nlm.nih.gov/pubmed/35898251?tool=bestpractice.com
Evidências de um ensaio randomizado e duplo-cego sugerem que os IBPs e os antagonistas H2 têm eficácia similar na redução do risco de hemorragia digestiva alta ou de úlceras em pessoas que tomam aspirina em baixas doses.[44]Chan FK, Kyaw M, Tanigawa T, et al. Similar efficacy of proton-pump inhibitors vs H2-receptor antagonists in reducing risk of upper gastrointestinal bleeding or ulcers in high-risk users of low-dose aspirin. Gastroenterology. 2016 Sep 15;152(1):105-10.e1.
http://www.ncbi.nlm.nih.gov/pubmed/27641510?tool=bestpractice.com
Uma metanálise que avaliou antagonistas H2, IBPs e análogos da prostaglandina constatou que os IBPs foram mais eficazes para prevenir o sangramento de úlcera que os antagonistas H2 e os análogos da prostaglandina.[45]Scally B, Emberson JR, Spata E, et al. Effects of gastroprotectant drugs for the prevention and treatment of peptic ulcer disease and its complications: a meta-analysis of randomised trials. Lancet Gastroenterol Hepatol. 2018 Apr;3(4):231-41.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5842491
http://www.ncbi.nlm.nih.gov/pubmed/29475806?tool=bestpractice.com
Os IBPs também foram mais eficazes para curar úlceras e prevenir o sangramento recorrente e a necessidade de transfusão de sangue.[45]Scally B, Emberson JR, Spata E, et al. Effects of gastroprotectant drugs for the prevention and treatment of peptic ulcer disease and its complications: a meta-analysis of randomised trials. Lancet Gastroenterol Hepatol. 2018 Apr;3(4):231-41.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5842491
http://www.ncbi.nlm.nih.gov/pubmed/29475806?tool=bestpractice.com