Aspirin and other nonsteroidal anti-inflammatory drugs (NSAIDs) should be used with caution, especially in people aged over 60 years and those who are taking corticosteroids, bisphosphonates, or other antithrombotic drugs.[24]García Rodríguez LA, Lin KJ, Hernández-Díaz S, et al. Risk of upper gastrointestinal bleeding with low-dose acetylsalicylic acid alone and in combination with clopidogrel and other medications. Circulation. 2011 Mar 15;123(10):1108-15.
https://www.ahajournals.org/doi/10.1161/CIRCULATIONAHA.110.973008?url_ver=Z39.88-2003&rfr_id=ori:rid:crossref.org&rfr_dat=cr_pub%20%200pubmed
http://www.ncbi.nlm.nih.gov/pubmed/21357821?tool=bestpractice.com
[25]Knopp-Sihota JA, Cummings GG, Homik J, et al. The association between serious upper gastrointestinal bleeding and incident bisphosphonate use: a population-based nested cohort study. BMC Geriatr. 2013 Apr 20;13:36.
https://bmcgeriatr.biomedcentral.com/articles/10.1186/1471-2318-13-36
http://www.ncbi.nlm.nih.gov/pubmed/23602075?tool=bestpractice.com
Concurrent use of a proton-pump inhibitor (PPI) has been shown to reduce the risk of gastrointestinal (GI) complications in patients taking long-term aspirin therapy and/or oral anticoagulants.[35]Scheiman JM, Devereaux PJ, Herlitz J, et al. Prevention of peptic ulcers with esomeprazole
in patients at risk of ulcer development treated with low-dose acetylsalicylic
acid: a randomised, controlled trial (OBERON). Heart. 2011 May;97(10):797-802.
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3088470/?tool=pubmed
http://www.ncbi.nlm.nih.gov/pubmed/21415072?tool=bestpractice.com
[36]Kurlander JE, Barnes GD, Fisher A, et al. Association of antisecretory drugs with upper gastrointestinal bleeding in patients using oral anticoagulants: a systematic review and meta-analysis. Am J Med. 2022 Oct;135(10):1231-43.e8.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10031639
http://www.ncbi.nlm.nih.gov/pubmed/35679879?tool=bestpractice.com
[37]Ahn HJ, Lee SR, Choi EK, et al. Protective effect of proton-pump inhibitor against gastrointestinal bleeding in patients receiving oral anticoagulants: a systematic review and meta-analysis. Br J Clin Pharmacol. 2022 Nov;88(11):4676-87.
http://www.ncbi.nlm.nih.gov/pubmed/35921204?tool=bestpractice.com
PPIs prevent peptic ulcers and complications in people who require NSAID therapy.[38]Yang M, He M, Zhao M, et al. Proton pump inhibitors for preventing non-steroidal anti-inflammatory drug induced gastrointestinal toxicity: a systematic review. Curr Med Res Opin. 2017 Jan 25;33(6):973-80.
http://www.ncbi.nlm.nih.gov/pubmed/28076696?tool=bestpractice.com
However, guidelines suggest considering a test and treat strategy for Helicobacter pyloribefore starting long-term NSAID therapy, as H pylori eradication has been shown to protect against aspirin-associated peptic ulcer bleeding.[33]Lanza FL, Chan FK, Quigley EM; Practice Parameters Committee of the American College of Gastroenterology. Guidelines for prevention of NSAID-related ulcer complications. Am J Gastroenterol. 2009 Mar;104(3):728-38.
http://www.ncbi.nlm.nih.gov/pubmed/19240698?tool=bestpractice.com
[39]Hawkey C, Avery A, Coupland CAC, et al. Helicobacter pylori eradication for primary prevention of peptic ulcer bleeding in older patients prescribed aspirin in primary care (HEAT): a randomised, double-blind, placebo-controlled trial. Lancet. 2022 Nov 5;400(10363):1597-606.
https://www.thelancet.com/journals/lancet/article/PIIS0140-6736(22)01843-8/fulltext
http://www.ncbi.nlm.nih.gov/pubmed/36335970?tool=bestpractice.com
PPI therapy may be more effective than misoprostol (a prostaglandin E1 analog) for the prevention of GI ulcers in people prescribed long-term NSAID therapy.
[
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Do misoprostol, H2-receptor antagonists, or proton pump inhibitors used for at least 12 weeks prevent upper gastrointestinal ulcers in patients requiring chronic NSAID use?/cca.html?targetUrl=https://cochranelibrary.com/cca/doi/10.1002/cca.430/fullShow me the answer Compliance with misoprostol (particularly at high doses) may be compromised by GI adverse effects, including abdominal cramping and diarrhea.
Prophylactic use of a PPI is appropriate for patients in intensive care, who are deemed at high risk of GI bleeding due comorbidities such as chronic liver disease, or have coexisting conditions such as coagulopathy, shock, or liver disease.[34]MacLaren R, Dionne JC, Granholm A, et al. Society of Critical Care Medicine and American Society of Health-System Pharmacists Guideline for the prevention of stress-related gastrointestinal bleeding in critically ill adults. Crit Care Med. 2024 Aug 1;52(8):e421-30.
https://journals.lww.com/ccmjournal/fulltext/2024/08000/society_of_critical_care_medicine_and_american.22.aspx
http://www.ncbi.nlm.nih.gov/pubmed/39007578?tool=bestpractice.com
[40]Cash BD. Evidence-based medicine as it applies to acid suppression in the hospitalized patient. Crit Care Med. 2002 Jun;30(suppl 6):S373-8.
http://www.ncbi.nlm.nih.gov/pubmed/12072665?tool=bestpractice.com
Mechanical ventilation by itself is no longer considered a risk factor.[34]MacLaren R, Dionne JC, Granholm A, et al. Society of Critical Care Medicine and American Society of Health-System Pharmacists Guideline for the prevention of stress-related gastrointestinal bleeding in critically ill adults. Crit Care Med. 2024 Aug 1;52(8):e421-30.
https://journals.lww.com/ccmjournal/fulltext/2024/08000/society_of_critical_care_medicine_and_american.22.aspx
http://www.ncbi.nlm.nih.gov/pubmed/39007578?tool=bestpractice.com
[41]Mutlu GM, Mutlu EA, Factor P. Prevention and treatment of gastrointestinal complications in patients on mechanical ventilation. Am J Respir Med. 2003;2(5):395-411.
http://www.ncbi.nlm.nih.gov/pubmed/14719992?tool=bestpractice.com
All critically ill adults with factors that likely increase the risk for stress-related upper GI bleeding should receive either a PPI or a H2 antagonists to prevent bleeding.[42]Reynolds PM, MacLaren R. Re-evaluating the utility of stress ulcer prophylaxis in the critically ill patient: a clinical scenario-based meta-analysis. Pharmacotherapy. 2019 Mar;39(3):408-20.
http://www.ncbi.nlm.nih.gov/pubmed/30101529?tool=bestpractice.com
[34]MacLaren R, Dionne JC, Granholm A, et al. Society of Critical Care Medicine and American Society of Health-System Pharmacists Guideline for the prevention of stress-related gastrointestinal bleeding in critically ill adults. Crit Care Med. 2024 Aug 1;52(8):e421-30.
https://journals.lww.com/ccmjournal/fulltext/2024/08000/society_of_critical_care_medicine_and_american.22.aspx
http://www.ncbi.nlm.nih.gov/pubmed/39007578?tool=bestpractice.com
Prophylaxis should be discontinued when critical illness is no longer evident or the risk factor(s) is no longer present despite ongoing critical illness.[34]MacLaren R, Dionne JC, Granholm A, et al. Society of Critical Care Medicine and American Society of Health-System Pharmacists Guideline for the prevention of stress-related gastrointestinal bleeding in critically ill adults. Crit Care Med. 2024 Aug 1;52(8):e421-30.
https://journals.lww.com/ccmjournal/fulltext/2024/08000/society_of_critical_care_medicine_and_american.22.aspx
http://www.ncbi.nlm.nih.gov/pubmed/39007578?tool=bestpractice.com
Discontinuation of stress ulcer prophylaxis before transfer out of the intensive care unit is necessary to prevent inappropriate prescribing.[43]Jones CA, Betthauser KD, Lizza BD, et al. Impact of stress ulcer prophylaxis discontinuation guidance in mechanically ventilated, critically ill patients: a pre-post cohort study. Hosp Pharm. 2022 Aug;57(4):510-7.
https://pmc.ncbi.nlm.nih.gov/articles/PMC9310319
http://www.ncbi.nlm.nih.gov/pubmed/35898251?tool=bestpractice.com
Evidence from one double-blind randomized trial suggests that PPIs and H2 antagonists have similar efficacy in reducing the risk of upper GI or ulcers in people taking low-dose aspirin.[44]Chan FK, Kyaw M, Tanigawa T, et al. Similar efficacy of proton-pump inhibitors vs H2-receptor antagonists in reducing risk of upper gastrointestinal bleeding or ulcers in high-risk users of low-dose aspirin. Gastroenterology. 2016 Sep 15;152(1):105-10.e1.
http://www.ncbi.nlm.nih.gov/pubmed/27641510?tool=bestpractice.com
A meta-analysis that evaluated H2 antagonists, PPIs, and prostaglandin analogs found that PPIs were more effective in preventing bleeding from ulcers than H2 antagonists and prostaglandin analogs.[45]Scally B, Emberson JR, Spata E, et al. Effects of gastroprotectant drugs for the prevention and treatment of peptic ulcer disease and its complications: a meta-analysis of randomised trials. Lancet Gastroenterol Hepatol. 2018 Apr;3(4):231-41.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5842491
http://www.ncbi.nlm.nih.gov/pubmed/29475806?tool=bestpractice.com
PPIs were also more effective in healing ulcers and preventing recurrent bleeding and the need for blood transfusion.[45]Scally B, Emberson JR, Spata E, et al. Effects of gastroprotectant drugs for the prevention and treatment of peptic ulcer disease and its complications: a meta-analysis of randomised trials. Lancet Gastroenterol Hepatol. 2018 Apr;3(4):231-41.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5842491
http://www.ncbi.nlm.nih.gov/pubmed/29475806?tool=bestpractice.com