Patients with JIA, or suspected JIA, should be managed by a specialist paediatric rheumatology multidisciplinary team.[57]Davies K, Cleary G, Foster H, et al. BSPAR Standards of Care for children and young people with juvenile idiopathic arthritis. Rheumatology (Oxford). 2010 Jul;49(7):1406-8.
https://academic.oup.com/rheumatology/article/49/7/1406/1785261/BSPAR-Standards-of-Care-for-children-and-young
http://www.ncbi.nlm.nih.gov/pubmed/20173199?tool=bestpractice.com
The goals of treatment are:
Achieving clinically inactive disease
Excellent symptom control
Prevention and minimisation of of joint damage
Prevention and minimisation of treatment side effects
Promotion of good physical and mental health.
Prompt initiation of disease-modifying therapy is essential, because active, uncontrolled JIA can cause permanent joint damage.[58]Ringold S, Angeles-Han ST, Beukelman T, et al. 2019 American College of Rheumatology/Arthritis Foundation guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for non-systemic polyarthritis, sacroiliitis, and enthesitis. Arthritis Care Res (Hoboken). 2019 Jun;71(6):717-34.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6561125
http://www.ncbi.nlm.nih.gov/pubmed/31021516?tool=bestpractice.com
Specific therapy is indicated by disease phenotype, disease activity, and presence/absence of risk factors.
Phenotypic groups
The treatment of JIA varies according to the predominant clinical features. American College of Rheumatology (ACR) guidelines define treatment groups by clinical phenotype rather than International League of Associations for Rheumatology categories. The patient groups are:[58]Ringold S, Angeles-Han ST, Beukelman T, et al. 2019 American College of Rheumatology/Arthritis Foundation guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for non-systemic polyarthritis, sacroiliitis, and enthesitis. Arthritis Care Res (Hoboken). 2019 Jun;71(6):717-34.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6561125
http://www.ncbi.nlm.nih.gov/pubmed/31021516?tool=bestpractice.com
[59]Beukelman T, Patkar NM, Saag KG, et al. 2011 American College of Rheumatology recommendations for the treatment of juvenile idiopathic arthritis: initiation and safety monitoring of therapeutic agents for the treatment of arthritis and systemic features. Arthritis Care Res (Hoboken). 2011 Apr;63(4):465-82.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3222233
http://www.ncbi.nlm.nih.gov/pubmed/21452260?tool=bestpractice.com
Patients with psoriatic arthritis may belong to the polyarticular JIA, sacroiliitis, or enthesitis phenotypic group.[58]Ringold S, Angeles-Han ST, Beukelman T, et al. 2019 American College of Rheumatology/Arthritis Foundation guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for non-systemic polyarthritis, sacroiliitis, and enthesitis. Arthritis Care Res (Hoboken). 2019 Jun;71(6):717-34.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6561125
http://www.ncbi.nlm.nih.gov/pubmed/31021516?tool=bestpractice.com
Assessing disease activity
Disease activity is assessed by:
Each of these four factors is a component of the Juvenile Arthritis Disease Activity Score.[60]Consolaro A, Ruperto N, Bazso A, et al. Development and validation of a composite disease activity score for juvenile idiopathic arthritis. Arthritis Rheum. 2009 May 15;61(5):658-66.
https://onlinelibrary.wiley.com/doi/10.1002/art.24516
http://www.ncbi.nlm.nih.gov/pubmed/19405003?tool=bestpractice.com
Disease activity scores can help the clinician select an appropriate initial treatment, and recognise a need to escalate treatment.
Physician and patient global assessment of disease activity is performed using a Likert scale. The physician rates the disease activity from 0 (no activity) to 10 (maximum activity). The patient (or parent) rates patient wellbeing from 0 (very good) to 10 (very poor).[61]Consolaro A, Giancane G, Schiappapietra B, et al. Clinical outcome measures in juvenile idiopathic arthritis. Pediatr Rheumatol Online J. 2016 Apr 18;14(1):23.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4836071
http://www.ncbi.nlm.nih.gov/pubmed/27089922?tool=bestpractice.com
A joint is considered active if it is swollen or has limited motion with pain/tenderness.
Low disease activity is not the same as disease remission, and should prompt a re-evaluation of therapy.
Supportive care
All aspects of the child’s physical and psychological health should be evaluated and addressed by the multidisciplinary team.[57]Davies K, Cleary G, Foster H, et al. BSPAR Standards of Care for children and young people with juvenile idiopathic arthritis. Rheumatology (Oxford). 2010 Jul;49(7):1406-8.
https://academic.oup.com/rheumatology/article/49/7/1406/1785261/BSPAR-Standards-of-Care-for-children-and-young
http://www.ncbi.nlm.nih.gov/pubmed/20173199?tool=bestpractice.com
Physiotherapy and occupational therapy are recommended for children with, or at risk of, functional limitations.[58]Ringold S, Angeles-Han ST, Beukelman T, et al. 2019 American College of Rheumatology/Arthritis Foundation guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for non-systemic polyarthritis, sacroiliitis, and enthesitis. Arthritis Care Res (Hoboken). 2019 Jun;71(6):717-34.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6561125
http://www.ncbi.nlm.nih.gov/pubmed/31021516?tool=bestpractice.com
Patients should be encouraged to participate in interests, sport, and community life.[57]Davies K, Cleary G, Foster H, et al. BSPAR Standards of Care for children and young people with juvenile idiopathic arthritis. Rheumatology (Oxford). 2010 Jul;49(7):1406-8.
https://academic.oup.com/rheumatology/article/49/7/1406/1785261/BSPAR-Standards-of-Care-for-children-and-young
http://www.ncbi.nlm.nih.gov/pubmed/20173199?tool=bestpractice.com
Inactivity leads to deconditioning and disability.[62]Long AR, Rouster-Stevens KA. The role of exercise therapy in the management of juvenile idiopathic arthritis. Curr Opin Rheumatol. 2010 Mar;22(2):213-7.
http://www.ncbi.nlm.nih.gov/pubmed/20010296?tool=bestpractice.com
Weight-bearing activity may reduce the risk of low bone mineral density.[63]Gannotti ME, Nahorniak M, Gorton GE III, et al. Can exercise influence low bone mineral density in children with juvenile rheumatoid arthritis? Pediatr Phys Ther. 2007 Summer;19(2):128-39.
http://www.ncbi.nlm.nih.gov/pubmed/17505290?tool=bestpractice.com
One Cochrane review found that exercise therapy does not appear to increase quality of life, exercise capacity, functional ability, or pain in patients with JIA; neither is it associated with any adverse effects or exacerbation of arthritis. However, heterogeneous outcome measures were used in the included trials, and the authors suggest that more standardised outcome measures are needed to evaluate the long-term effect of exercise therapy.[64]Takken T, van Brussel M, Engelbert RH, et al. Exercise therapy in juvenile idiopathic arthritis. Cochrane Database Syst Rev. 2008 Apr 16;(2):CD005954.
https://www.cochranelibrary.com/cdsr/doi/10.1002/14651858.CD005954.pub2/full
http://www.ncbi.nlm.nih.gov/pubmed/18425929?tool=bestpractice.com
Foot orthoses may reduce pain and improve quality of life in children with JIA.[65]Coda A, Fowlie PW, Davidson JE, et al. Foot orthoses in children with juvenile idiopathic arthritis: a randomised controlled trial. Arch Dis Child. 2014 Jul;99(7):649-51.
http://www.ncbi.nlm.nih.gov/pubmed/24636956?tool=bestpractice.com
[66]Brosseau L, Toupin-April K, Wells G, et al. Ottawa Panel evidence-based clinical practice guidelines for foot care in the management of juvenile idiopathic arthritis. Arch Phys Med Rehabil. 2016 Jul;97(7):1163-81.
http://www.ncbi.nlm.nih.gov/pubmed/26707409?tool=bestpractice.com
Patients with JIA have an increased risk of psychiatric morbidity.[67]Mullick MS, Nahar JS, Haq SA. Psychiatric morbidity, stressors, impact, and burden in juvenile idiopathic arthritis. J Health Popul Nutr. 2005 Jun;23(2):142-9.
http://www.ncbi.nlm.nih.gov/pubmed/16117366?tool=bestpractice.com
Support and strategies for managing any difficulties should be provided.[57]Davies K, Cleary G, Foster H, et al. BSPAR Standards of Care for children and young people with juvenile idiopathic arthritis. Rheumatology (Oxford). 2010 Jul;49(7):1406-8.
https://academic.oup.com/rheumatology/article/49/7/1406/1785261/BSPAR-Standards-of-Care-for-children-and-young
http://www.ncbi.nlm.nih.gov/pubmed/20173199?tool=bestpractice.com
Polyarticular JIA
Conventional synthetic disease-modifying antirheumatic drugs (DMARDs) include methotrexate, sulfasalazine, and leflunomide.
Methotrexate is first-line initial therapy for children with polyarticular JIA.[58]Ringold S, Angeles-Han ST, Beukelman T, et al. 2019 American College of Rheumatology/Arthritis Foundation guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for non-systemic polyarthritis, sacroiliitis, and enthesitis. Arthritis Care Res (Hoboken). 2019 Jun;71(6):717-34.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6561125
http://www.ncbi.nlm.nih.gov/pubmed/31021516?tool=bestpractice.com
Randomised controlled trials have demonstrated improvement in joint symptoms and a reduction in disease activity with methotrexate.[68]Ruperto N, Murray KJ, Gerloni V, et al. A randomized trial of parenteral methotrexate comparing an intermediate dose with a higher dose in children with juvenile idiopathic arthritis who failed to respond to standard doses of methotrexate. Arthritis Rheum. 2004 Jul;50(7):2191-201.
http://www.ncbi.nlm.nih.gov/pubmed/15248217?tool=bestpractice.com
[69]Giannini EH, Brewer EJ, Kuzmina N, et al. Methotrexate in resistant juvenile rheumatoid arthritis. Results of the U.S.A.-U.S.S.R. double-blind, placebo-controlled trial. N Engl J Med. 1992 Apr 16;326(16):1043-9.
http://www.ncbi.nlm.nih.gov/pubmed/1549149?tool=bestpractice.com
Folic acid is usually given concomitantly to decrease the side effects of methotrexate, and anti-emetics may be used to reduce nausea. Patients should be counselled to avoid alcohol and pregnancy while taking methotrexate.
Full blood count, serum creatinine, and liver enzymes should be checked before starting methotrexate, and every 3 to 4 months during treatment.[70]Onel KB, Horton DB, Lovell DJ, et al. 2021 American College of Rheumatology guideline for the treatment of juvenile idiopathic arthritis: recommendations for nonpharmacologic therapies, medication monitoring, immunizations, and imaging. Arthritis Care Res (Hoboken). 2022 Apr;74(4):505-20.
http://www.ncbi.nlm.nih.gov/pubmed/35233989?tool=bestpractice.com
Patients at risk of hepatitis B or hepatitis C infection should have a screening antibody test before starting methotrexate.[59]Beukelman T, Patkar NM, Saag KG, et al. 2011 American College of Rheumatology recommendations for the treatment of juvenile idiopathic arthritis: initiation and safety monitoring of therapeutic agents for the treatment of arthritis and systemic features. Arthritis Care Res (Hoboken). 2011 Apr;63(4):465-82.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3222233
http://www.ncbi.nlm.nih.gov/pubmed/21452260?tool=bestpractice.com
Elevation of aspartate aminotransferase (AST) or alanine aminotransferase (ALT) above 2 times the upper limit justifies temporary suspension of methotrexate, which can be re-started following normalisation of serum liver enzyme levels.[59]Beukelman T, Patkar NM, Saag KG, et al. 2011 American College of Rheumatology recommendations for the treatment of juvenile idiopathic arthritis: initiation and safety monitoring of therapeutic agents for the treatment of arthritis and systemic features. Arthritis Care Res (Hoboken). 2011 Apr;63(4):465-82.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3222233
http://www.ncbi.nlm.nih.gov/pubmed/21452260?tool=bestpractice.com
Some trials have demonstrated the safety and efficacy of leflunomide as a second-line conventional synthetic DMARD in paediatric patients who are intolerant or unresponsive to methotrexate. Most of the paediatric patients responsive to leflunomide maintained their response in a 2-year open-label extension study.[71]Silverman E, Mouy R, Spiegel L, et al. Leflunomide or methotrexate for juvenile rheumatoid arthritis. N Engl J Med. 2005 Apr 21;352(16):1655-66.
http://www.nejm.org/doi/full/10.1056/NEJMoa041810#t=article
http://www.ncbi.nlm.nih.gov/pubmed/15843668?tool=bestpractice.com
Sulfasalazine may also be used as a second-line option.[58]Ringold S, Angeles-Han ST, Beukelman T, et al. 2019 American College of Rheumatology/Arthritis Foundation guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for non-systemic polyarthritis, sacroiliitis, and enthesitis. Arthritis Care Res (Hoboken). 2019 Jun;71(6):717-34.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6561125
http://www.ncbi.nlm.nih.gov/pubmed/31021516?tool=bestpractice.com
Biological therapies that block the action of inflammatory cytokines, including tumour necrosis factor (TNF)-alpha, interleukin (IL)-1, and IL-6, are highly effective and have revolutionised the treatment of JIA. These therapies are typically given in addition to a DMARD. They may be given as part of initial therapy in patients with risk factors for a poor prognosis, or started after an inadequate response to a conventional synthetic DMARD.[58]Ringold S, Angeles-Han ST, Beukelman T, et al. 2019 American College of Rheumatology/Arthritis Foundation guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for non-systemic polyarthritis, sacroiliitis, and enthesitis. Arthritis Care Res (Hoboken). 2019 Jun;71(6):717-34.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6561125
http://www.ncbi.nlm.nih.gov/pubmed/31021516?tool=bestpractice.com
Risk factors for poor prognosis include:[58]Ringold S, Angeles-Han ST, Beukelman T, et al. 2019 American College of Rheumatology/Arthritis Foundation guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for non-systemic polyarthritis, sacroiliitis, and enthesitis. Arthritis Care Res (Hoboken). 2019 Jun;71(6):717-34.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6561125
http://www.ncbi.nlm.nih.gov/pubmed/31021516?tool=bestpractice.com
Presence of anti-cyclic citrullinated peptide antibodies
Presence of rheumatoid factor
Joint damage at presentation
High-risk joint involvement (cervical spine, wrist, or hip)
High disease activity
Patient judged by physician to be at high risk of disabling joint damage.
A TNF-alpha inhibitor is first-line.[58]Ringold S, Angeles-Han ST, Beukelman T, et al. 2019 American College of Rheumatology/Arthritis Foundation guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for non-systemic polyarthritis, sacroiliitis, and enthesitis. Arthritis Care Res (Hoboken). 2019 Jun;71(6):717-34.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6561125
http://www.ncbi.nlm.nih.gov/pubmed/31021516?tool=bestpractice.com
Treatment with etanercept or adalimumab is preferred to treatment with infliximab. Infliximab is given by intravenous infusion and carries a risk of infusion-associated reactions and is not approved for the treatment of any form of JIA.
Etanercept is a soluble TNF-alpha receptor antagonist. It is approved for polyarticular disease in children 2 years of age and over.[72]Lovell DJ, Giannini EH, Reiff A, et al. Etanercept in children with polyarticular juvenile rheumatoid arthritis. N Engl J Med. 2000 Mar 16;342(11):763-9.
http://www.nejm.org/doi/full/10.1056/NEJM200003163421103#t=article
http://www.ncbi.nlm.nih.gov/pubmed/10717011?tool=bestpractice.com
An open-label extension trial has demonstrated safety and efficacy for up to 8 years of use.[73]Lovell DJ, Reiff A, Ilowite NT, et al. Safety and efficacy of up to eight years of continuous etanercept therapy in patients with juvenile rheumatoid arthritis. Arthritis Rheum. 2008 May;58(5):1496-504.
http://www.ncbi.nlm.nih.gov/pubmed/18438876?tool=bestpractice.com
Adalimumab is a recombinant humanised TNF-alpha inhibitor that is approved for polyarticular disease in children 2 years of age and over.[74]Lovell DJ, Ruperto N, Goodman S, et al. Adalimumab with or without methotrexate in juvenile rheumatoid arthritis. N Engl J Med. 2008 Aug 21;359(8):810-20.
http://www.nejm.org/doi/full/10.1056/NEJMoa0706290#t=article
http://www.ncbi.nlm.nih.gov/pubmed/18716298?tool=bestpractice.com
Over 70% of children receiving adalimumab in combination with methotrexate had a 70% improvement in at least three of the ACR core set variables after 16 weeks of therapy.[74]Lovell DJ, Ruperto N, Goodman S, et al. Adalimumab with or without methotrexate in juvenile rheumatoid arthritis. N Engl J Med. 2008 Aug 21;359(8):810-20.
http://www.nejm.org/doi/full/10.1056/NEJMoa0706290#t=article
http://www.ncbi.nlm.nih.gov/pubmed/18716298?tool=bestpractice.com
It is also effective in patients with enthesitis.[75]Burgos-Vargas R, Tse SM, Horneff G, et al. A randomized, double-blind, placebo-controlled multicenter study of adalimumab in pediatric patients with enthesitis-related arthritis. Arthritis Care Res (Hoboken). 2015 Nov;67(11):1503-12.
http://onlinelibrary.wiley.com/doi/10.1002/acr.22657/full
http://www.ncbi.nlm.nih.gov/pubmed/26223543?tool=bestpractice.com
The long-term tolerability and efficacy of adalimumab in JIA has been demonstrated.[76]Klotsche J, Niewerth M, Haas JP, et al. Long-term safety of etanercept and adalimumab compared to methotrexate in patients with juvenile idiopathic arthritis (JIA). Ann Rheum Dis. 2016 May;75(5):855-61.
http://www.ncbi.nlm.nih.gov/pubmed/25926155?tool=bestpractice.com
[77]Lovell DJ, Brunner HI, Reiff AO, et al. Long-term outcomes in patients with polyarticular juvenile idiopathic arthritis receiving adalimumab with or without methotrexate. RMD Open. 2020 Jul;6(2):e001208.
https://rmdopen.bmj.com/content/6/2/e001208.long
http://www.ncbi.nlm.nih.gov/pubmed/32665432?tool=bestpractice.com
Infliximab is a monoclonal, chimeric TNF-alpha inhibitor.[78]Ruperto N, Lovell DJ, Cuttica R, et al. A randomized, placebo-controlled trial of infliximab plus methotrexate for the treatment of polyarticular-course juvenile rheumatoid arthritis. Arthritis Rheum. 2007 Sep;56(9):3096-106.
http://www.ncbi.nlm.nih.gov/pubmed/17763439?tool=bestpractice.com
Monoclonal antibodies have analogies to murine proteins, meaning pre-medication with antihistamines, paracetamol, and corticosteroids is advised to minimise infusion-associated reactions.[79]Aeschlimann FA, Hofer KD, Cannizzaro Schneider E, et al. Infliximab in pediatric rheumatology patients: a retrospective analysis of infusion reactions and severe adverse events during 2246 infusions over 12 years. J Rheumatol. 2014 Jul;41(7):1409-15.
https://www.jrheum.org/content/41/7/1409.long
http://www.ncbi.nlm.nih.gov/pubmed/24833759?tool=bestpractice.com
[80]Bartoli F, Bruni C, Cometi L, et al. Premedication prevents infusion reactions and improves retention rate during infliximab treatment. Clin Rheumatol. 2016 Nov;35(11):2841-5.
http://www.ncbi.nlm.nih.gov/pubmed/27436188?tool=bestpractice.com
TNF-alpha inhibitors should be used with caution in patients with recurrent infections, conditions predisposing to infections, pre-existing demyelinating disorders, or haematological diseases, due to the immunosuppressive nature of these medicines.[81]Carrasco R, Smith JA, Lovell D. Biologic agents for the treatment of juvenile rheumatoid arthritis. Paediatr Drugs. 2004;6(3):137-46.
http://www.ncbi.nlm.nih.gov/pubmed/15170361?tool=bestpractice.com
A study evaluating etanercept and adalimumab showed an increase in number of infections but no clear evidence that the overall malignancy risk was increased.[76]Klotsche J, Niewerth M, Haas JP, et al. Long-term safety of etanercept and adalimumab compared to methotrexate in patients with juvenile idiopathic arthritis (JIA). Ann Rheum Dis. 2016 May;75(5):855-61.
http://www.ncbi.nlm.nih.gov/pubmed/25926155?tool=bestpractice.com
Chronic carriers of tuberculosis and hepatitis B are susceptible to disease reactivation. Tuberculosis skin tests, and viral hepatitis screening for patients with risk factors for infection, are recommended prior to treatment.[59]Beukelman T, Patkar NM, Saag KG, et al. 2011 American College of Rheumatology recommendations for the treatment of juvenile idiopathic arthritis: initiation and safety monitoring of therapeutic agents for the treatment of arthritis and systemic features. Arthritis Care Res (Hoboken). 2011 Apr;63(4):465-82.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3222233
http://www.ncbi.nlm.nih.gov/pubmed/21452260?tool=bestpractice.com
[81]Carrasco R, Smith JA, Lovell D. Biologic agents for the treatment of juvenile rheumatoid arthritis. Paediatr Drugs. 2004;6(3):137-46.
http://www.ncbi.nlm.nih.gov/pubmed/15170361?tool=bestpractice.com
Live vaccines should be avoided during treatment.[82]Yokota S, Mori M, Imagawa T, et al. Guidelines on the use of etanercept for juvenile idiopathic arthritis in Japan. Mod Rheumatol. 2010 Apr;20(2):107-13.
http://www.ncbi.nlm.nih.gov/pubmed/20087751?tool=bestpractice.com
Tocilizumab (an IL-6 inhibitor) or abatacept (a fusion protein) are used if the patient does not respond to a TNF-alpha inhibitor.
Tocilizumab can be used as monotherapy or in combination with methotrexate for children with polyarticular JIA. Tocilizumab is relatively well tolerated and has proven efficacy for up to 52 weeks.[83]Schoels MM, van der Heijde D, Breedveld FC, et al. Blocking the effects of interleukin-6 in rheumatoid arthritis and other inflammatory rheumatic diseases: systematic literature review and meta-analysis informing a consensus statement. Ann Rheum Dis. 2013 Apr;72(4):583-9.
http://ard.bmj.com/content/72/4/583.long
http://www.ncbi.nlm.nih.gov/pubmed/23144446?tool=bestpractice.com
It is approved in children 2 years of age and older.
Serious hepatotoxicity (including acute liver failure, hepatitis, and jaundice) has been identified in eight patients treated with tocilizumab worldwide. Two patients required liver transplantation. Serious liver injury has been reported from 2 weeks to more than 5 years after starting treatment. While liver toxicity occurs rarely and the risk-benefit profile still supports the use of tocilizumab, the ACR recommends monitoring ALT or AST at initiation of treatment, within 4 to 8 weeks of treatment and every 3 to 4 months thereafter.[70]Onel KB, Horton DB, Lovell DJ, et al. 2021 American College of Rheumatology guideline for the treatment of juvenile idiopathic arthritis: recommendations for nonpharmacologic therapies, medication monitoring, immunizations, and imaging. Arthritis Care Res (Hoboken). 2022 Apr;74(4):505-20.
http://www.ncbi.nlm.nih.gov/pubmed/35233989?tool=bestpractice.com
Be cautious when considering starting tocilizumab treatment in patients with ALT or AST levels higher than 1.5 times the upper limit of normal. Tocilizumab is not recommended if ALT or AST levels are higher than 5 times the upper limit of normal. If liver enzyme abnormalities are identified, consider a dose modification (reduction, interruption, or discontinuation) according to the manufacturer’s recommendations. Advise patients to seek medical help immediately if they experience signs and symptoms of hepatic injury.[84]Medicines and Healthcare products Regulatory Agency. Tocilizumab (RoActemra): rare risk of serious liver injury including cases requiring transplantation. July 2019 [internet publication].
https://www.gov.uk/drug-safety-update/tocilizumab-roactemra-rare-risk-of-serious-liver-injury-including-cases-requiring-transplantation
Abatacept is a recombinant, fully humanised fusion protein composed of the extracellular domain of human CTLA-4 and a portion of the Fc-domain of human immunoglobulin G-1. It is used in children aged 2 years and older with polyarticular JIA who have had an inadequate response to previous conventional synthetic DMARDs, and has proven efficacy and long-term safety.[85]Ruperto N, Lovell DJ, Quartier P, et al. Abatacept in children with juvenile idiopathic arthritis: a randomised, double-blind, placebo-controlled withdrawal trial. Lancet. 2008 Aug 2;372(9636):383-91.
http://www.ncbi.nlm.nih.gov/pubmed/18632147?tool=bestpractice.com
[86]Ruperto N, Lovell DJ, Quartier P, et al. Long-term safety and efficacy of abatacept in children with juvenile idiopathic arthritis. Arthritis Rheum. 2010 Jun;62(6):1792-802.
http://onlinelibrary.wiley.com/doi/10.1002/art.27431/full
http://www.ncbi.nlm.nih.gov/pubmed/20191582?tool=bestpractice.com
[87]European Medicines Agency. Summary of opinion (post authorisation): Orencia - abatacept. January 2019 [internet publication].
https://www.ema.europa.eu/en/documents/smop/chmp-post-authorisation-summary-positive-opinion-orencia-x-117-g_en.pdf
Improvements in health-related quality of life were observed during a phase 3, double-blind, placebo controlled trial with abatacept, providing real-life, tangible benefits to children with JIA and their parents or carers.[88]Ruperto N, Lovell DJ, Li T, et al. Abatacept improves health-related quality of life, pain, sleep quality, and daily participation in subjects with juvenile idiopathic arthritis. Arthritis Care Res. 2010 Nov;62(11):1542-51.
http://onlinelibrary.wiley.com/doi/10.1002/acr.20283/full
http://www.ncbi.nlm.nih.gov/pubmed/20597110?tool=bestpractice.com
Non-steroidal anti-inflammatory drugs (NSAIDs) are used as adjunctive therapy to treat pain and stiffness in children with polyarticular JIA while systemic therapies take effect.
Specific NSAIDs are approved for children with JIA (e.g., ibuprofen, naproxen, meloxicam). Others are commonly used off-label. No specific NSAID is superior to another.[89]Eccleston C, Cooper TE, Fisher E, et al. Non-steroidal anti-inflammatory drugs (NSAIDs) for chronic non-cancer pain in children and adolescents. Cochrane Database Syst Rev. 2017 Aug 2;8(8):CD012537.
https://www.cochranelibrary.com/cdsr/doi/10.1002/14651858.CD012537.pub2/full
http://www.ncbi.nlm.nih.gov/pubmed/28770976?tool=bestpractice.com
Sequential trials of different NSAIDs are used to identify the most effective medicine for individual patients.
Possible adverse effects include renal impairment, gastrointestinal symptoms (nausea, constipation, diarrhoea, abdominal pain), headache, and rash.[89]Eccleston C, Cooper TE, Fisher E, et al. Non-steroidal anti-inflammatory drugs (NSAIDs) for chronic non-cancer pain in children and adolescents. Cochrane Database Syst Rev. 2017 Aug 2;8(8):CD012537.
https://www.cochranelibrary.com/cdsr/doi/10.1002/14651858.CD012537.pub2/full
http://www.ncbi.nlm.nih.gov/pubmed/28770976?tool=bestpractice.com
Low-dose oral corticosteroid therapy can be used for up to 3 months to improve symptoms while systemic therapies take effect. This treatment is particularly helpful for children with polyarticular JIA with high or moderate disease activity.[46]Ringold S, Weiss PF, Beukelman T, et al. 2013 update of the 2011 American College of Rheumatology recommendations for the treatment of juvenile idiopathic arthritis: recommendations for the medical therapy of children with systemic juvenile idiopathic arthritis and tuberculosis screening among children receiving biologic medications. Arthritis Rheum. 2013 Oct;65(10):2499-512.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5408575
http://www.ncbi.nlm.nih.gov/pubmed/24092554?tool=bestpractice.com
Intra-articular corticosteroid injections can be used alone or as part of a treatment plan involving other systemic treatments. Radiographical assistance may be necessary for injecting some joints. The procedure can be undertaken with the administration of entonox or general anaesthetic to the child.
Relief is expected to last for at least 4 months.[59]Beukelman T, Patkar NM, Saag KG, et al. 2011 American College of Rheumatology recommendations for the treatment of juvenile idiopathic arthritis: initiation and safety monitoring of therapeutic agents for the treatment of arthritis and systemic features. Arthritis Care Res (Hoboken). 2011 Apr;63(4):465-82.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3222233
http://www.ncbi.nlm.nih.gov/pubmed/21452260?tool=bestpractice.com
Injections can be repeated every 4 months as needed. Adverse effects from intra-articular injections are uncommon.
Intra-articular corticosteroid injections may not be a suitable treatment for large numbers of joints that have been injected multiple times. Escalation of systemic therapy may be more appropriate.[58]Ringold S, Angeles-Han ST, Beukelman T, et al. 2019 American College of Rheumatology/Arthritis Foundation guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for non-systemic polyarthritis, sacroiliitis, and enthesitis. Arthritis Care Res (Hoboken). 2019 Jun;71(6):717-34.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6561125
http://www.ncbi.nlm.nih.gov/pubmed/31021516?tool=bestpractice.com
Duration of relief <4 months may also imply a need to escalate systemic therapy.[59]Beukelman T, Patkar NM, Saag KG, et al. 2011 American College of Rheumatology recommendations for the treatment of juvenile idiopathic arthritis: initiation and safety monitoring of therapeutic agents for the treatment of arthritis and systemic features. Arthritis Care Res (Hoboken). 2011 Apr;63(4):465-82.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3222233
http://www.ncbi.nlm.nih.gov/pubmed/21452260?tool=bestpractice.com
Oligoarticular JIA
Corticosteroid injections are first-line treatment for most patients.[59]Beukelman T, Patkar NM, Saag KG, et al. 2011 American College of Rheumatology recommendations for the treatment of juvenile idiopathic arthritis: initiation and safety monitoring of therapeutic agents for the treatment of arthritis and systemic features. Arthritis Care Res (Hoboken). 2011 Apr;63(4):465-82.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3222233
http://www.ncbi.nlm.nih.gov/pubmed/21452260?tool=bestpractice.com
Initial NSAID monotherapy may be given for 2 months if the child has low disease activity, no contractures, and no poor prognostic features, to relieve joint pain and swelling.[59]Beukelman T, Patkar NM, Saag KG, et al. 2011 American College of Rheumatology recommendations for the treatment of juvenile idiopathic arthritis: initiation and safety monitoring of therapeutic agents for the treatment of arthritis and systemic features. Arthritis Care Res (Hoboken). 2011 Apr;63(4):465-82.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3222233
http://www.ncbi.nlm.nih.gov/pubmed/21452260?tool=bestpractice.com
Poor prognostic features are:[59]Beukelman T, Patkar NM, Saag KG, et al. 2011 American College of Rheumatology recommendations for the treatment of juvenile idiopathic arthritis: initiation and safety monitoring of therapeutic agents for the treatment of arthritis and systemic features. Arthritis Care Res (Hoboken). 2011 Apr;63(4):465-82.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3222233
http://www.ncbi.nlm.nih.gov/pubmed/21452260?tool=bestpractice.com
Arthritis of the hip or cervical spine
Arthritis of the ankle or wrist plus prolonged or marked inflammatory marker elevation
Radiographic evidence of erosions or joint space narrowing.
If there is any residual disease activity after 2 months’ treatment, therapy should be escalated to intra-articular corticosteroid injections.[59]Beukelman T, Patkar NM, Saag KG, et al. 2011 American College of Rheumatology recommendations for the treatment of juvenile idiopathic arthritis: initiation and safety monitoring of therapeutic agents for the treatment of arthritis and systemic features. Arthritis Care Res (Hoboken). 2011 Apr;63(4):465-82.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3222233
http://www.ncbi.nlm.nih.gov/pubmed/21452260?tool=bestpractice.com
Methotrexate is used if a patient has not responded to intra-articular corticosteroids, or as initial treatment for children with high disease activity and adverse prognostic features.[59]Beukelman T, Patkar NM, Saag KG, et al. 2011 American College of Rheumatology recommendations for the treatment of juvenile idiopathic arthritis: initiation and safety monitoring of therapeutic agents for the treatment of arthritis and systemic features. Arthritis Care Res (Hoboken). 2011 Apr;63(4):465-82.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3222233
http://www.ncbi.nlm.nih.gov/pubmed/21452260?tool=bestpractice.com
TNF-alpha inhibitors are rarely needed for patients with oligoarticular JIA, but they should be considered in patients with ongoing active disease despite treatment with intra-articular corticosteroids and methotrexate.[59]Beukelman T, Patkar NM, Saag KG, et al. 2011 American College of Rheumatology recommendations for the treatment of juvenile idiopathic arthritis: initiation and safety monitoring of therapeutic agents for the treatment of arthritis and systemic features. Arthritis Care Res (Hoboken). 2011 Apr;63(4):465-82.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3222233
http://www.ncbi.nlm.nih.gov/pubmed/21452260?tool=bestpractice.com
When treatment with a TNF-alpha inhibitor is needed, etanercept or adalimumab are preferred to infliximab. Infliximab is given by intravenous infusion and carries a risk of infusion-associated reactions and is not approved for the treatment of any form of JIA.
Sacroiliitis
First-line treatment is NSAID monotherapy. Oral corticosteroids may be used to relieve symptoms for up to 3 months during initiation or escalation of systemic therapy.[58]Ringold S, Angeles-Han ST, Beukelman T, et al. 2019 American College of Rheumatology/Arthritis Foundation guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for non-systemic polyarthritis, sacroiliitis, and enthesitis. Arthritis Care Res (Hoboken). 2019 Jun;71(6):717-34.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6561125
http://www.ncbi.nlm.nih.gov/pubmed/31021516?tool=bestpractice.com
Treatment should be escalated to a TNF-alpha inhibitor if disease activity is not controlled by NSAID monotherapy. Use of TNF-alpha inhibitors is associated with decreased disease activity, compared with placebo.[90]Horneff G, Fitter S, Foeldvari I, et al. Double-blind, placebo-controlled randomized trial with adalimumab for treatment of juvenile onset ankylosing spondylitis (JoAS): significant short term improvement. Arthritis Res Ther. 2012 Oct 24;14(5):R230.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3580542
http://www.ncbi.nlm.nih.gov/pubmed/23095307?tool=bestpractice.com
[91]Hugle B, Burgos-Vargas R, Inman RD, et al. Long-term outcome of anti-tumor necrosis factor alpha blockade in the treatment of juvenile spondyloarthritis. Clin Exp Rheumatol. 2014 May-Jun;32(3):424-31.
http://www.ncbi.nlm.nih.gov/pubmed/24387974?tool=bestpractice.com
[92]Horneff G, Burgos-Vargas R, Constantin T, et al. Efficacy and safety of open-label etanercept on extended oligoarticular juvenile idiopathic arthritis, enthesitis-related arthritis and psoriatic arthritis: part 1 (week 12) of the CLIPPER study. Ann Rheum Dis. 2014 Jun;73(6):1114-22.
https://ard.bmj.com/content/73/6/1114.long
http://www.ncbi.nlm.nih.gov/pubmed/23696632?tool=bestpractice.com
Treatment with etanercept or adalimumab is preferred to treatment with infliximab. Infliximab is given by intravenous infusion and carries a risk of infusion-associated reactions and is not approved for the treatment of any form of JIA.
Sulfasalazine may be used instead of a TNF-alpha inhibitor, particularly for children in whom TNF-alpha inhibitors are contraindicated or not tolerated.[58]Ringold S, Angeles-Han ST, Beukelman T, et al. 2019 American College of Rheumatology/Arthritis Foundation guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for non-systemic polyarthritis, sacroiliitis, and enthesitis. Arthritis Care Res (Hoboken). 2019 Jun;71(6):717-34.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6561125
http://www.ncbi.nlm.nih.gov/pubmed/31021516?tool=bestpractice.com
Enthesitis
First-line treatment is NSAID monotherapy. Oral corticosteroids may be used to relieve symptoms for up to 3 months during initiation or escalation of systemic therapy.[58]Ringold S, Angeles-Han ST, Beukelman T, et al. 2019 American College of Rheumatology/Arthritis Foundation guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for non-systemic polyarthritis, sacroiliitis, and enthesitis. Arthritis Care Res (Hoboken). 2019 Jun;71(6):717-34.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6561125
http://www.ncbi.nlm.nih.gov/pubmed/31021516?tool=bestpractice.com
Treatment should be escalated if there is active enthesitis despite NSAID monotherapy.[58]Ringold S, Angeles-Han ST, Beukelman T, et al. 2019 American College of Rheumatology/Arthritis Foundation guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for non-systemic polyarthritis, sacroiliitis, and enthesitis. Arthritis Care Res (Hoboken). 2019 Jun;71(6):717-34.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6561125
http://www.ncbi.nlm.nih.gov/pubmed/31021516?tool=bestpractice.com
Typically methotrexate or sulfasalazine are used first, with escalation to a TNF-alpha inhibitor if the child doesn’t respond.[93]Mistry RR, Patro P, Agarwal V, et al. Enthesitis-related arthritis: current perspectives. Open Access Rheumatol. 2019 Jan 25;11:19-31.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6354696
http://www.ncbi.nlm.nih.gov/pubmed/30774484?tool=bestpractice.com
When treatment with a TNF-alpha inhibitor is required, etanercept or adalimumab are preferred to infliximab. Infliximab is given by intravenous infusion and carries a risk of infusion-associated reactions and is not approved for the treatment of any form of JIA.
However, the ACR guidelines recommend that children with active enthesitis despite NSAID monotherapy should escalate to TNF-alpha inhibitors, rather than methotrexate or sulfasalazine, and noted that the level of evidence for this recommendation was low.[58]Ringold S, Angeles-Han ST, Beukelman T, et al. 2019 American College of Rheumatology/Arthritis Foundation guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for non-systemic polyarthritis, sacroiliitis, and enthesitis. Arthritis Care Res (Hoboken). 2019 Jun;71(6):717-34.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6561125
http://www.ncbi.nlm.nih.gov/pubmed/31021516?tool=bestpractice.com
One observational study reported a greater improvement in pain and disease activity after 12 months in children with enthesitis who received a TNF-alpha inhibitor, compared with those who received a DMARD alone.[94]Weiss PF, Xiao R, Brandon TG, et al. Comparative effectiveness of tumor necrosis factor agents and disease-modifying antirheumatic therapy in children with enthesitis-related arthritis: the first year after diagnosis. J Rheumatol. 2018 Jan;45(1):107-14.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5750113
http://www.ncbi.nlm.nih.gov/pubmed/28916542?tool=bestpractice.com
Systemic-onset JIA
The ACR recommends that the management of systemic JIA is based on a confirmed diagnosis of JIA and whether it has features of macrophage activation syndrome (MAS).[95]Onel KB, Horton DB, Lovell DJ, et al. 2021 American College of Rheumatology guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for oligoarthritis, temporomandibular joint arthritis, and systemic juvenile idiopathic arthritis. Arthritis Care Res (Hoboken). 2022 Apr;74(4):521-37.
http://www.ncbi.nlm.nih.gov/pubmed/35233986?tool=bestpractice.com
MAS is a life-threatening complication of systemic-onset JIA. Signs and symptoms include:[96]Shakoory B, Geerlinks A, Wilejto M, et al. The 2022 EULAR/ACR points to consider at the early stages of diagnosis and management of suspected haemophagocytic lymphohistiocytosis/macrophage activation syndrome (HLH/MAS). Ann Rheum Dis. 2023 Oct;82(10):1271-85.
https://ard.bmj.com/content/82/10/1271.long
http://www.ncbi.nlm.nih.gov/pubmed/37487610?tool=bestpractice.com
Persistent fever
Elevated and/or rising ferritin or other markers of inflammation/damage
Inappropriately low or declining haemoglobin, platelet counts or white blood cells (neutrophils and lymphocytes)
Hepatic dysfunction
Coagulopathy
Splenomegaly
Central nervous system dysfunction
About 10% to 15% of patients with systemic-onset JIA develop life-threatening overt MAS.[97]Schulert GS, Yasin S, Carey B, et al. Systemic juvenile idiopathic arthritis-associated lung disease: characterization and risk factors. Arthritis Rheumatol. 2019 Nov;71(11):1943-54.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6817389
http://www.ncbi.nlm.nih.gov/pubmed/31379071?tool=bestpractice.com
MAS is present if the following criteria are met in a febrile patient with known or suspected systemic-onset JIA: ferritin >684 micrograms/L (>684 ng/mL) and any two of platelet count ≤181 x 10⁹/L, aspartate aminotransferase >48 U/L, triglycerides >1.76 mmol/L (>156 mg/dL), or fibrinogen ≤3.6 g/L (≤360 mg/dL).[98]Ravelli A, Minoia F, Davì S, et al. 2016 classification criteria for macrophage activation syndrome complicating systemic juvenile idiopathic arthritis: a European League Against Rheumatism/American College of Rheumatology/Paediatric Rheumatology International Trials Organisation Collaborative initiative. Arthritis Rheumatol. 2016 Mar;68(3):566-76.
https://onlinelibrary.wiley.com/doi/10.1002/art.39332
http://www.ncbi.nlm.nih.gov/pubmed/26314788?tool=bestpractice.com
If a patient has a normal ferritin level, but there is ongoing clinical suspicion of MAS, serial ferritin testing should be considered.[96]Shakoory B, Geerlinks A, Wilejto M, et al. The 2022 EULAR/ACR points to consider at the early stages of diagnosis and management of suspected haemophagocytic lymphohistiocytosis/macrophage activation syndrome (HLH/MAS). Ann Rheum Dis. 2023 Oct;82(10):1271-85.
https://ard.bmj.com/content/82/10/1271.long
http://www.ncbi.nlm.nih.gov/pubmed/37487610?tool=bestpractice.com
Consult a paediatric rheumatology specialist urgently if features of MAS are present. Patients with MAS can deteriorate rapidly and may require intensive care admission. For patients with suspected MAS, initiating treatment while diagnostic testing is in progress should be considered.[96]Shakoory B, Geerlinks A, Wilejto M, et al. The 2022 EULAR/ACR points to consider at the early stages of diagnosis and management of suspected haemophagocytic lymphohistiocytosis/macrophage activation syndrome (HLH/MAS). Ann Rheum Dis. 2023 Oct;82(10):1271-85.
https://ard.bmj.com/content/82/10/1271.long
http://www.ncbi.nlm.nih.gov/pubmed/37487610?tool=bestpractice.com
Monitoring initial treatment response by assessing clinical and laboratory markers of organ involvement should be assessed at least daily, and markers of systemic inflammation at least twice weekly. Worsening or lack of improvement in laboratory parameters of systemic inflammation, particularly ferritin, may indicate disease progression and a need to reassess diagnosis and/or treatment.[96]Shakoory B, Geerlinks A, Wilejto M, et al. The 2022 EULAR/ACR points to consider at the early stages of diagnosis and management of suspected haemophagocytic lymphohistiocytosis/macrophage activation syndrome (HLH/MAS). Ann Rheum Dis. 2023 Oct;82(10):1271-85.
https://ard.bmj.com/content/82/10/1271.long
http://www.ncbi.nlm.nih.gov/pubmed/37487610?tool=bestpractice.com
The ACR recommends early use of biological agents in children with systemic JIA due to their proven effectiveness, moving away from former recommendations that focused on corticosteroids and conventional synthetic DMARDs.
Systemic JIA without MAS
Initial treatment is with a biological agent (i.e., IL-1 or IL-6 inhibitor) and/or an NSAID.[95]Onel KB, Horton DB, Lovell DJ, et al. 2021 American College of Rheumatology guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for oligoarthritis, temporomandibular joint arthritis, and systemic juvenile idiopathic arthritis. Arthritis Care Res (Hoboken). 2022 Apr;74(4):521-37.
http://www.ncbi.nlm.nih.gov/pubmed/35233986?tool=bestpractice.com
There is some evidence that those with systemic JIA without MAS will respond to NSAIDs alone and even have clinically inactive disease.[95]Onel KB, Horton DB, Lovell DJ, et al. 2021 American College of Rheumatology guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for oligoarthritis, temporomandibular joint arthritis, and systemic juvenile idiopathic arthritis. Arthritis Care Res (Hoboken). 2022 Apr;74(4):521-37.
http://www.ncbi.nlm.nih.gov/pubmed/35233986?tool=bestpractice.com
Patients who undergo an initial trial of NSAID monotherapy should be followed up within 2 weeks for evaluation of a possible need for drug escalation.[99]Sura A, Failing C, Sturza J, et al. Patient characteristics associated with response to NSAID monotherapy in children with systemic juvenile idiopathic arthritis. Pediatr Rheumatol Online J. 2018 Jan 5;16(1):2.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5755314
http://www.ncbi.nlm.nih.gov/pubmed/29304824?tool=bestpractice.com
If a response occurs and inactive disease occurs, then NSAIDs should be tapered and discontinued. If clinical response is not rapid and complete, rapid escalation of therapy is recommended. Several NSAIDs are approved for children with JIA (e.g., ibuprofen, naproxen, meloxicam). Others are commonly used off-label. No specific NSAID is superior to another.[89]Eccleston C, Cooper TE, Fisher E, et al. Non-steroidal anti-inflammatory drugs (NSAIDs) for chronic non-cancer pain in children and adolescents. Cochrane Database Syst Rev. 2017 Aug 2;8(8):CD012537.
https://www.cochranelibrary.com/cdsr/doi/10.1002/14651858.CD012537.pub2/full
http://www.ncbi.nlm.nih.gov/pubmed/28770976?tool=bestpractice.com
Sequential trials of different NSAIDs are used to identify the most effective drug for individual patients. Possible adverse effects include renal impairment, gastrointestinal symptoms, headache, and rash.[89]Eccleston C, Cooper TE, Fisher E, et al. Non-steroidal anti-inflammatory drugs (NSAIDs) for chronic non-cancer pain in children and adolescents. Cochrane Database Syst Rev. 2017 Aug 2;8(8):CD012537.
https://www.cochranelibrary.com/cdsr/doi/10.1002/14651858.CD012537.pub2/full
http://www.ncbi.nlm.nih.gov/pubmed/28770976?tool=bestpractice.com
Biological agents can be given in combination with an NSAID for initial treatment or after a trial period of an NSAID. The ACR does not recommend any one preferred agent, but indicates that IL-1 inhibitors (e.g., anakinra, canakinumab) and IL-6 inhibitors (e.g., tocilizumab) are extremely effective and well-tolerated options. The choice should be based on discussions between the practitioner and patient as routes of administration and frequency vary. The ACR recommends switching between IL-1 and IL-6 inhibitors when needed due to a lack of efficacy or poor tolerability as individual response varies significantly.[95]Onel KB, Horton DB, Lovell DJ, et al. 2021 American College of Rheumatology guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for oligoarthritis, temporomandibular joint arthritis, and systemic juvenile idiopathic arthritis. Arthritis Care Res (Hoboken). 2022 Apr;74(4):521-37.
http://www.ncbi.nlm.nih.gov/pubmed/35233986?tool=bestpractice.com
[100]Tarp S, Amarilyo G, Foeldvari I, et al. Efficacy and safety of biological agents for systemic juvenile idiopathic arthritis: a systematic review and meta-analysis of randomized trials. Rheumatology (Oxford). 2016 Apr;55(4):669-79.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5854101
http://www.ncbi.nlm.nih.gov/pubmed/26628580?tool=bestpractice.com
[101]Ruperto N, Brunner HI, Quartier P, et al; PRINTO; PRCSG. Two randomized trials of canakinumab in systemic juvenile idiopathic arthritis. N Engl J Med. 2012 Dec 20;367(25):2396-406.
http://www.nejm.org/doi/full/10.1056/NEJMoa1205099#t=article
http://www.ncbi.nlm.nih.gov/pubmed/23252526?tool=bestpractice.com
[102]Pascual V, Allantaz F, Arce E, et al. Role of interleukin-1 (IL-1) in the pathogenesis of systemic onset juvenile idiopathic arthritis and clinical response to IL-1 blockade. J Exp Med. 2005 May 2;201(9):1479-86.
https://rupress.org/jem/article/201/9/1479/46269/Role-of-interleukin-1-IL-1-in-the-pathogenesis-of
http://www.ncbi.nlm.nih.gov/pubmed/15851489?tool=bestpractice.com
Biological agents used in systemic JIA appear safe and comparable with respect to adverse effect risk in the short term.[100]Tarp S, Amarilyo G, Foeldvari I, et al. Efficacy and safety of biological agents for systemic juvenile idiopathic arthritis: a systematic review and meta-analysis of randomized trials. Rheumatology (Oxford). 2016 Apr;55(4):669-79.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5854101
http://www.ncbi.nlm.nih.gov/pubmed/26628580?tool=bestpractice.com
Anakinra has a short half-life, meaning its dose can be adjusted or it can be withdrawn quickly. One randomised controlled trial reported a response rate of 66% to 1 month's treatment with anakinra, compared with 8% to placebo, in children with systemic JIA. After 1 month, 83% of the children receiving placebo were switched to anakinra; 90% of children who switched from placebo responded to anakinra.[103]Quartier P, Allantaz F, Cimaz R, et al. A multicentre, randomised, double-blind, placebo-controlled trial with the interleukin-1 receptor antagonist anakinra in patients with systemic-onset juvenile idiopathic arthritis (ANAJIS trial). Ann Rheum Dis. 2011 May;70(5):747-54.
https://ard.bmj.com/content/70/5/747.long
http://www.ncbi.nlm.nih.gov/pubmed/21173013?tool=bestpractice.com
Canakinumab is effective for treating active systemic JIA.[101]Ruperto N, Brunner HI, Quartier P, et al; PRINTO; PRCSG. Two randomized trials of canakinumab in systemic juvenile idiopathic arthritis. N Engl J Med. 2012 Dec 20;367(25):2396-406.
http://www.nejm.org/doi/full/10.1056/NEJMoa1205099#t=article
http://www.ncbi.nlm.nih.gov/pubmed/23252526?tool=bestpractice.com
[104]Brunner HI, Quartier P, Alexeeva E, et al. Efficacy and safety of canakinumab in patients with systemic juvenile idiopathic arthritis with and without fever at baseline: results from an open-label, active-treatment extension study. Arthritis Rheumatol. 2020 Dec;72(12):2147-58.
http://www.ncbi.nlm.nih.gov/pubmed/32648697?tool=bestpractice.com
Treatment with canakinumab significantly reduces fever and disease activity, compared with placebo.[101]Ruperto N, Brunner HI, Quartier P, et al; PRINTO; PRCSG. Two randomized trials of canakinumab in systemic juvenile idiopathic arthritis. N Engl J Med. 2012 Dec 20;367(25):2396-406.
http://www.nejm.org/doi/full/10.1056/NEJMoa1205099#t=article
http://www.ncbi.nlm.nih.gov/pubmed/23252526?tool=bestpractice.com
One randomised trial showed a significant reduction in fever and active arthritis in children with systemic JIA refractory to corticosteroids and NSAIDs who were treated with tocilizumab, compared with placebo.[105]De Benedetti F, Brunner HI, Ruperto N, et al. Randomized trial of tocilizumab in systemic juvenile idiopathic arthritis. N Engl J Med. 2012 Dec 20;367(25):2385-95.
https://www.nejm.org/doi/10.1056/NEJMoa1112802
http://www.ncbi.nlm.nih.gov/pubmed/23252525?tool=bestpractice.com
Meta-analysis has shown similar efficacy between tocilizumab, canakinumab, and anakinra.[100]Tarp S, Amarilyo G, Foeldvari I, et al. Efficacy and safety of biological agents for systemic juvenile idiopathic arthritis: a systematic review and meta-analysis of randomized trials. Rheumatology (Oxford). 2016 Apr;55(4):669-79.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5854101
http://www.ncbi.nlm.nih.gov/pubmed/26628580?tool=bestpractice.com
One meta analysis of randomised controlled trials found that canakinumab had the highest probability of being the best treatment, in terms of the modified ACR Pediatric 30 (ACRpedi30) response rate, followed by anakinra and tocilizumab.[106]Song GG, Lee YH. Comparison of the efficacy and safety of biological agents in patients with systemic juvenile idiopathic arthritis: a Bayesian network meta-analysis of randomized controlled trials. Int J Clin Pharmacol Ther. 2021 Mar;59(3):239-46.
http://www.ncbi.nlm.nih.gov/pubmed/33191906?tool=bestpractice.com
Serious hepatotoxicity (including acute liver failure, hepatitis, and jaundice) has been identified with tocilizumab. The ACR recommends monitoring ALT or AST at initiation of treatment, within 4 to 8 weeks of treatment and every 3 to 4 months thereafter.[70]Onel KB, Horton DB, Lovell DJ, et al. 2021 American College of Rheumatology guideline for the treatment of juvenile idiopathic arthritis: recommendations for nonpharmacologic therapies, medication monitoring, immunizations, and imaging. Arthritis Care Res (Hoboken). 2022 Apr;74(4):505-20.
http://www.ncbi.nlm.nih.gov/pubmed/35233989?tool=bestpractice.com
Be cautious when considering starting tocilizumab treatment in patients with ALT or AST levels higher than 1.5 times the upper limit of normal. Tocilizumab is not recommended if ALT or AST levels are higher than 5 times the upper limit of normal. If liver enzyme abnormalities are identified, consider a dose modification (reduction, interruption, or discontinuation) according to the manufacturer’s recommendations.[84]Medicines and Healthcare products Regulatory Agency. Tocilizumab (RoActemra): rare risk of serious liver injury including cases requiring transplantation. July 2019 [internet publication].
https://www.gov.uk/drug-safety-update/tocilizumab-roactemra-rare-risk-of-serious-liver-injury-including-cases-requiring-transplantation
A range of small-scale trials demonstrated resolution of systemic signs following the use of biological agents.[103]Quartier P, Allantaz F, Cimaz R, et al. A multicentre, randomised, double-blind, placebo-controlled trial with the interleukin-1 receptor antagonist anakinra in patients with systemic-onset juvenile idiopathic arthritis (ANAJIS trial). Ann Rheum Dis. 2011 May;70(5):747-54.
https://ard.bmj.com/content/70/5/747.long
http://www.ncbi.nlm.nih.gov/pubmed/21173013?tool=bestpractice.com
[105]De Benedetti F, Brunner HI, Ruperto N, et al. Randomized trial of tocilizumab in systemic juvenile idiopathic arthritis. N Engl J Med. 2012 Dec 20;367(25):2385-95.
https://www.nejm.org/doi/10.1056/NEJMoa1112802
http://www.ncbi.nlm.nih.gov/pubmed/23252525?tool=bestpractice.com
[107]Ruperto N, Quartier P, Wulffraat N, et al. A phase II, multicenter, open-label study evaluating dosing and preliminary safety and efficacy of canakinumab in systemic juvenile idiopathic arthritis with active systemic features. Arthritis Rheum. 2012 Feb;64(2):557-67.
https://onlinelibrary.wiley.com/doi/epdf/10.1002/art.33342
http://www.ncbi.nlm.nih.gov/pubmed/21953497?tool=bestpractice.com
[108]Lovell DJ, Giannini EH, Reiff AO, et al. Long-term safety and efficacy of rilonacept in patients with systemic juvenile idiopathic arthritis. Arthritis Rheum. 2013 Sep;65(9):2486-96.
https://onlinelibrary.wiley.com/doi/epdf/10.1002/art.38042
http://www.ncbi.nlm.nih.gov/pubmed/23754188?tool=bestpractice.com
With prolonged use, some patients suffered from adverse effects (e.g., infection, neutropenia, and increased aminotransferase levels).[105]De Benedetti F, Brunner HI, Ruperto N, et al. Randomized trial of tocilizumab in systemic juvenile idiopathic arthritis. N Engl J Med. 2012 Dec 20;367(25):2385-95.
https://www.nejm.org/doi/10.1056/NEJMoa1112802
http://www.ncbi.nlm.nih.gov/pubmed/23252525?tool=bestpractice.com
The ACR recommends considering tapering and discontinuing biological therapies when the disease is deemed inactive.[95]Onel KB, Horton DB, Lovell DJ, et al. 2021 American College of Rheumatology guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for oligoarthritis, temporomandibular joint arthritis, and systemic juvenile idiopathic arthritis. Arthritis Care Res (Hoboken). 2022 Apr;74(4):521-37.
http://www.ncbi.nlm.nih.gov/pubmed/35233986?tool=bestpractice.com
Conventional synthetic DMARDs in combination with biological agents can be considered in people with an inadequate response.
Systemic JIA with MAS
Initial treatment includes a biological agent and/or corticosteroid.[95]Onel KB, Horton DB, Lovell DJ, et al. 2021 American College of Rheumatology guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for oligoarthritis, temporomandibular joint arthritis, and systemic juvenile idiopathic arthritis. Arthritis Care Res (Hoboken). 2022 Apr;74(4):521-37.
http://www.ncbi.nlm.nih.gov/pubmed/35233986?tool=bestpractice.com
Biological agent monotherapy may not be sufficient for severely ill patients. Biological agents combined with a corticosteroid and a conventional synthetic DMARD may be necessary to control MAS in some patients.[95]Onel KB, Horton DB, Lovell DJ, et al. 2021 American College of Rheumatology guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for oligoarthritis, temporomandibular joint arthritis, and systemic juvenile idiopathic arthritis. Arthritis Care Res (Hoboken). 2022 Apr;74(4):521-37.
http://www.ncbi.nlm.nih.gov/pubmed/35233986?tool=bestpractice.com
If a combination is used, then it is typically continued until disease control is established. If a patient is receiving both a biological agent or conventional synthetic DMARD and a corticosteroid, the corticosteroid should be tapered and discontinued first before attempting to taper the biological agent or the conventional synthetic DMARD. It is unclear how soon or rapidly these can be safely discontinued in patients with inactive systemic JIA.[95]Onel KB, Horton DB, Lovell DJ, et al. 2021 American College of Rheumatology guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for oligoarthritis, temporomandibular joint arthritis, and systemic juvenile idiopathic arthritis. Arthritis Care Res (Hoboken). 2022 Apr;74(4):521-37.
http://www.ncbi.nlm.nih.gov/pubmed/35233986?tool=bestpractice.com
Although there are potential effects on bone health and growth, corticosteroids are conditionally recommended by the ACR as part of the initial treatment of acute systemic JIA with MAS.[95]Onel KB, Horton DB, Lovell DJ, et al. 2021 American College of Rheumatology guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for oligoarthritis, temporomandibular joint arthritis, and systemic juvenile idiopathic arthritis. Arthritis Care Res (Hoboken). 2022 Apr;74(4):521-37.
http://www.ncbi.nlm.nih.gov/pubmed/35233986?tool=bestpractice.com
[109]Guzman J, Kerr T, Ward LM, et al. Growth and weight gain in children with juvenile idiopathic arthritis: results from the ReACCh-Out cohort. Pediatr Rheumatol Online J. 2017 Aug 22;15(1):68.
https://ped-rheum.biomedcentral.com/articles/10.1186/s12969-017-0196-7
http://www.ncbi.nlm.nih.gov/pubmed/28830457?tool=bestpractice.com
Glucocorticoid therapy should be limited to the lowest effective dose for the shortest duration possible, although treatment with high-dose corticosteroids may be required for initial disease control.[95]Onel KB, Horton DB, Lovell DJ, et al. 2021 American College of Rheumatology guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for oligoarthritis, temporomandibular joint arthritis, and systemic juvenile idiopathic arthritis. Arthritis Care Res (Hoboken). 2022 Apr;74(4):521-37.
http://www.ncbi.nlm.nih.gov/pubmed/35233986?tool=bestpractice.com
Long-term corticosteroid therapy in children is not appropriate because of its potential side effects on bone health and growth.[109]Guzman J, Kerr T, Ward LM, et al. Growth and weight gain in children with juvenile idiopathic arthritis: results from the ReACCh-Out cohort. Pediatr Rheumatol Online J. 2017 Aug 22;15(1):68.
https://ped-rheum.biomedcentral.com/articles/10.1186/s12969-017-0196-7
http://www.ncbi.nlm.nih.gov/pubmed/28830457?tool=bestpractice.com
Treatment with biological agents may mask some MAS features and lead to limitations in diagnosis.[110]Schulert GS, Minoia F, Bohnsack J, et al. Effect of biologic therapy on clinical and laboratory features of macrophage activation syndrome associated with systemic juvenile idiopathic arthritis. Arthritis Care Res (Hoboken). 2018 Mar;70(3):409-19.
https://onlinelibrary.wiley.com/doi/epdf/10.1002/acr.23277
http://www.ncbi.nlm.nih.gov/pubmed/28499329?tool=bestpractice.com
In children with systemic JIA whose disease is inactive, it may be possible to maintain this inactive disease state with lower doses of, or discontinuation of, biological agents.[111]Ter Haar NM, van Dijkhuizen EHP, Swart JF, et al. Treatment to target using recombinant interleukin-1 receptor antagonist as first-line monotherapy in new-onset systemic juvenile idiopathic arthritis: results from a five-year follow-up study. Arthritis Rheumatol. 2019 Jul;71(7):1163-73.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6617757
http://www.ncbi.nlm.nih.gov/pubmed/30848528?tool=bestpractice.com
[112]Quartier P, Alexeeva E, Constantin T, et al. Tapering canakinumab monotherapy in patients with systemic juvenile idiopathic arthritis in clinical remission: results from a phase IIIb/IV open-label, randomized study. Arthritis Rheumatol. 2021 Feb;73(2):336-46.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7898684
http://www.ncbi.nlm.nih.gov/pubmed/32783351?tool=bestpractice.com
Conventional synthetic DMARDs are strongly recommended over long-term corticosteroids for residual arthritis and incomplete response to IL-1 and/or IL-6 inhibitors.[95]Onel KB, Horton DB, Lovell DJ, et al. 2021 American College of Rheumatology guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for oligoarthritis, temporomandibular joint arthritis, and systemic juvenile idiopathic arthritis. Arthritis Care Res (Hoboken). 2022 Apr;74(4):521-37.
http://www.ncbi.nlm.nih.gov/pubmed/35233986?tool=bestpractice.com
There is no preferred agent.[95]Onel KB, Horton DB, Lovell DJ, et al. 2021 American College of Rheumatology guideline for the treatment of juvenile idiopathic arthritis: therapeutic approaches for oligoarthritis, temporomandibular joint arthritis, and systemic juvenile idiopathic arthritis. Arthritis Care Res (Hoboken). 2022 Apr;74(4):521-37.
http://www.ncbi.nlm.nih.gov/pubmed/35233986?tool=bestpractice.com
The primary conventional synthetic DMARD used for the treatment of systemic JIA is methotrexate. Methotrexate has been commonly used in children with systemic JIA due to its corticosteroid-sparing effect.[113]DeWitt EM, Kimura Y, Beukelman T, et al. Consensus treatment plans for new-onset systemic juvenile idiopathic arthritis. Arthritis Care Res (Hoboken). 2012 Jul;64(7):1001-10.
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3368104
http://www.ncbi.nlm.nih.gov/pubmed/22290637?tool=bestpractice.com
Although it is used less frequently, it can be given alone or alongside a biological agent to control symptoms. Leflunomide is another conventional synthetic DMARD that can be used in JIA to manage the inflammatory response when methotrexate is not tolerated.[71]Silverman E, Mouy R, Spiegel L, et al. Leflunomide or methotrexate for juvenile rheumatoid arthritis. N Engl J Med. 2005 Apr 21;352(16):1655-66.
http://www.nejm.org/doi/full/10.1056/NEJMoa041810#t=article
http://www.ncbi.nlm.nih.gov/pubmed/15843668?tool=bestpractice.com
[114]Foeldvari I, Wierk A. Effectiveness of leflunomide in patients with juvenile idiopathic arthritis in clinical practice. J Rheumatol. 2010 Aug 1;37(8):1763-7.
https://www.jrheum.org/content/37/8/1763.long
http://www.ncbi.nlm.nih.gov/pubmed/20472925?tool=bestpractice.com
Tacrolimus, ciclosporin, cyclophosphamide, etoposide, chlorambucil, and azathioprine have been used in the treatment of systemic JIA, but are used less frequently due to the introduction of biological agents.